戻る
「早戻しボタン」を押すと検索画面に戻ります。 [閉じる]

コーパス検索結果 (１語後でソート)

通し番号をクリックするとPubMedの該当ページを表示します
1  nucleophilic fragmentation of the resulting isoxazoline.
2 em and masking the twofold aldol motif as an isoxazoline.
3 ollowed by alkynyl addition to the resultant isoxazoline.
4 strategy to prepare chalcogen-functionalized isoxazolines.
5 e preparation of chiral 3,4,4-trisubstituted isoxazolines.
6 sfer reaction that leads to the formation of isoxazolines.
7  the synthesis of 3-substituted 5,5-dimethyl isoxazolines.
8 t state reactivity of oximes, specifically 2-isoxazolines.
9 ed [3+2] dipolar cycloaddition gave bicyclic isoxazoline 17 in a regio- and stereoselective fashion.
10 sulfonamide groups, in conjunction with (5R)-isoxazoline (2S)-diaminopropionate stereochemistry, were
11 t state reactivity of oximes, specifically 2-isoxazoline-3-carboxylates.
12 des with (meth-)acrylates into 3-substituted isoxazoline-5-carboxylates.
13 f antibacterial agents incorporating a novel isoxazoline A-ring surrogate.
14             The synthetic versatility of the isoxazoline allowed for a broad study of metal binding g
15          In a gratifying result, the initial isoxazoline analogue prepared was found to exhibit in vi
16  activity profile of a preliminary series of isoxazoline analogues incorporating either a C-C or N-C
17         Recently, we reported on a series of isoxazoline and isoxazole monobasic noncovalent inhibito
18                 Hence, the unification of an isoxazoline and peroxide heterocycles could be a potenti
19                                              Isoxazolines and 4-membered heterocycles are significant
20  synthesis of pyrrolidine-2-ylidenes from NH-isoxazolines and electron-deficient allenes.
21      The reaction of cyclic nitronic esters (isoxazoline- and 5,6-dihydro-4H-1,2-oxazine-N-oxides) wi
22                                    Using the isoxazoline as a common structural feature, three series
23 re a straightforward method employing chiral isoxazolines as key intermediates to access five differe
24       A novel synthetic route to spirocyclic isoxazolines based on a redox-neutral dearomative cycliz
25 observed between this series and a series of isoxazoline-based selective GPIIbIIIa antagonists.
26        Hydrogenolysis of C(5)-functionalized isoxazolines, bearing trimethylsilyl, phosphonate, or su
27 -pot synthesis of 3-substituted 5,5-dimethyl isoxazolines can be successfully achieved.
28   Alkaloid 6 contains a spirocyclohexadienyl-isoxazoline-carboxamide amide coupled to 2-aminohistamin
29 et of lotilaner, a synthetic molecule of the isoxazoline chemical class.
30 more stable and more synthetically versatile isoxazoline core.
31 ompounds, 3-phenyl-5-((phenylselanyl)methyl)-isoxazoline, demonstrated better anti-inflammatory and a
32                                           An isoxazoline derivative of [6]-gingerol was prepared and
33                       Cycloaddition provided isoxazoline derivative which upon hydrogenolysis furnish
34  report a series of novel biaryl-substituted isoxazoline derivatives in which the biaryl moiety was d
35 ria, by screening a small library of 3-bromo-isoxazoline derivatives that inactivate the enzyme throu
36           A practical synthesis of isoxazole/isoxazoline derivatives via Machetti-De Sarlo reaction u
37                 Herein we report a series of isoxazoline derivatives which are potent FXa inhibitors.
38 ing 1,3-aminoalcohol, 1,3-diol, oxetane, and isoxazoline derivatives.
39 ntly extended to the synthesis of 5 new (bis)isoxazoline ditellurides.
40                                   Nine of 17 isoxazolines, each incorporating a different potential m
41 road substrate scope and affords spirocyclic isoxazolines featuring novel substitution patterns compa
42 nitrile oxide and an olefin (22) to yield an isoxazoline followed by subsequent conversion into the g
43  the synthesis of 3-substituted 5,5-dimethyl isoxazolines from diversely functionalized chlorooximes
44                 The direct attachment of the isoxazoline functional group on the graphene surfaces pr
45 on with nitrile oxides to form metal-binding isoxazoline functional groups with high densities.
46 cation of the alpha-carbamate substituent of isoxazoline GPIIb/IIIa (alphaIIb beta3) antagonist DMP 7
47  series of saccharin/isoxazole and saccharin/isoxazoline hybrids were synthesized by 1,3-dipolar cycl
48 ng 19 new selenium- and tellurium-containing isoxazolines in good yields after 1 h at room temperatur
49 e cycloaddition, providing novel 5-hydroxy-2-isoxazolines in high chemical yield with high levels of
50 itrones to give highly substituted 4-nitro-4-isoxazolines in high yields.
51 m alkenes leading to the direct synthesis of isoxazolines in the presence of tert-butyl nitrite, quin
52                     The previously described isoxazoline inhibitor binds at the same site as DAP but
53 DAP) and a ternary complex with NADP+ and an isoxazoline inhibitor have been solved and refined again
54                    Grignard addition to this isoxazoline intermediate followed by DCC coupling of the
55 Protonation of the nitrogen of the metalated isoxazoline intermediate results in ring opening and the
56  electron transfer activation of the ensuing isoxazoline intermediate.
57 nocatalysis for the preparation of isoxazole/isoxazoline moieties in an environmentally benign fashio
58          The catalytic hydrogenolysis of the isoxazoline N-O bond was optimal upon using H(2) (1 atm)
59  which underwent N-O coupling to produce new isoxazoline N-oxide derivative.
60 oximes via one-pot halogenation/oxidation of isoxazoline N-oxide derivatives is described here.
61 romative cyclization of 3-benzyl-substituted isoxazoline N-oxides has been developed.
62                                The resulting isoxazoline N-oxides undergo catalytic reductive cleavag
63 ype recyclization of properly functionalized isoxazoline N-oxides was developed.
64                 In all cases, the respective isoxazoline products are produced with exquisite regio-
65 nes/alkenes to afford a library of isoxazole/isoxazoline products.
66 nitroso acetal, in which the N-O bond of the isoxazoline ring is selectively cleaved upon the action
67 side chain at the quaternary position of the isoxazoline ring led to SK549 which showed subnanomolar
68         The reaction likely proceeds through isoxazoline ring opening with generation of an unstable
69 nter, and reversal of the orientation of the isoxazoline ring resulted in lowered potency and/or dura
70 1-propene-1,3-sultone affords the respective isoxazoline-ring-fused heterobicyclic products in modera
71 ation sequence to access the C7 hydroxylated isoxazoline scaffold in one step and (2) a regioselectiv
72 alternative basic groups, elimination of the isoxazoline stereocenter, and reversal of the orientatio
73 zations of two styrenes are involved in this isoxazoline synthesis.
74  derivatives and trifluoromethylated benzo[c]isoxazoline systems, along with trifluoroacetyl nitrosob
75  novel class of peroxides containing a spiro-isoxazoline to primarily investigate the biological acti
76 ene, providing a comparable yield of desired isoxazolines under similar conditions.
77           We utilized 2 structurally related isoxazolines, which show in vitro inhibition of MIF taut
78                                        Using isoxazoline XR299 (1a) as a starting point for the desig