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1 f two moderately potent series of nonpeptide ETA receptor antagonists.
2 ides are potent and selective small molecule ETA receptor antagonists.
3 d this increase was blocked with a selective ET(A) receptor antagonist.
4 H compound of our series of novel synthetic (ET(A)) receptor antagonists.
5 n, either saline (negative control), BQ-123 (ETA receptor antagonist, 10 microg/min), BQ-788 (ETB rec
7 structural elements in a biphenylsulfonamide ET(A) receptor antagonist (2) followed by additional opt
8 ET-1 (2 and 6 pmol/min); BQ-123, a selective ET(A) receptor antagonist (3 and 10 nmol/min); and BQ-78
10 rteries of DOCA-salt rats with the selective ETA receptor antagonist ABT-627, NADPH oxidase inhibitor
11 ting our hypothesis that the combined use of ET(A) receptor antagonist (ABT-627; Atrasentan) with Tax
12 d DOCA-salt rats was reversed by a selective ET(A) receptor antagonist, ABT-627, the flavoprotein inh
13 e studied the effects of BQ 123, a selective ET(A) receptor antagonist, after ligation of the ductus
17 intravitreous injections of ET-1; BQ-123, an ETA receptor antagonist; and phosporamindon, an endothel
19 mized in a double-blind manner to either the ET(A) receptor antagonist atrasentan (10 mg) or placebo
20 oto-Kakizaki (GK) rats treated with vehicle, ET(A) receptor antagonist atrasentan (5 mg x kg(-1) x da
21 vels and that pretreatment with PD156707, an ETA receptor antagonist, blocks the rebound hypertension
23 vious exposure of cells to the endothelin-A (ET(A)) receptor antagonist BQ-123 (1 microm) prevented E
24 .001), whereas infusion of the endothelin-A (ET(A)) receptor antagonist BQ-123 significantly reduced
25 ium nitroprusside and the endothelin type A (ET(A)) receptor antagonist BQ-123 were assessed using ve
27 ne study, six subjects received placebo, the ETA receptor antagonist BQ-123 alone, and BQ-123 in comb
30 gonist, BQ-788, but not by the endothelin A (ET(A)) receptor antagonist, BQ-123, consistent with pred
31 ET-1-induced responses were inhibited by the ET(A) receptor antagonist BQ123 and the phospholipase C
33 ET1 effects on [Ca2+]i were prevented by the ETA receptor antagonist BQ123 (cyclo-D-Asp-Pro-D-Val-Leu
34 emia, we determined the effect of a specific ET(A) receptor antagonist, BQ123 (1mg/kg, intravenously
37 present study, we investigated the effect of ET(A) receptor antagonists, BQ123 and BMS182874, on morp
39 bation of coronary segments with a selective ETA receptor antagonist, BQ485 (1 mumol/L), had no effec
40 Et-1-induced IL-8 production was blocked by ET(A) receptor antagonist BQ610, but not by ET(B) recept
41 through ET(A) receptors, because a specific ET(A) receptor antagonist (BQ610) blocked these effects
42 by ET-1 was prevented by BQ-123, a selective ET(A) receptor antagonist, but was not affected by pertu
45 very of a potent and selective endothelin A (ETA) receptor antagonist for the potential treatment of
46 e Ad.ET-1 group, intravenous infusion of the ET(A) receptor antagonist FR 139317 reduced the blood pr
47 ion is therefore amenable to reversal by the ET(A) receptor antagonist FR139317, and this model may o
49 ith the infusion of either the endothelin-A (ETA) receptor antagonist FR139317, or saline vehicle.
51 at long-term treatment with an endothelin-A (ET(A)) receptor antagonist improves coronary endothelial
52 odynamic effects of sitaxsentan, a selective ET(A) receptor antagonist, in patients with chronic stab
53 tral endopeptidase inhibitor) and BQ-123 (an ETA receptor antagonist) increased FBF by 52 +/- 10% (P
56 We have previously disclosed the selective ET(A) receptor antagonist N-(3,4-dimethyl-5-isoxazolyl)-
57 during HPP (n=7), isch kidneys receiving the ETA receptor antagonist (n=7), and isch kidneys receivin
58 line, AngII infusion, AngII infusion with an ET(A) receptor antagonist, or AngII infusion with triple
60 concomitant administration of the selective ETA receptor antagonist (PD 156707 24 mg/d), and sham co
62 roteinuric CKD to compare the effects of the ET(A) receptor antagonist sitaxentan, nifedipine, and pl
63 n patients with HF, we infused the selective ET(A) receptor antagonist sitaxsentan at increasing rate
64 In a preliminary PAH study, the selective ET(A) receptor antagonist sitaxsentan improved six-min w
66 optimal dose of the selective endothelin A (ET(A)) receptor antagonist sitaxsentan for the treatment
67 osure to either BQ123 (10 microM), selective ETA receptor antagonist, U73122 (5 microM), or SKF 96365
69 dy, we show that HJP-272, a highly selective ET(A) receptor antagonist with an IC(50) of 70.1 nmol/L,
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