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1 mers were synthesized (N-aryl, N-alkyl and N-carbamate).
2 reaction of glycosylamines with fluorescent carbamate.
3 amines into well-ordered chains of ammonium carbamate.
4 ddition of CO2 since it cannot form a stable carbamate.
5 rting ADP and carbamoyl phosphate to ATP and carbamate.
6 ed by FTIR and tentatively assigned as a PTE carbamate.
7 and carbamoyl phosphate to ATP and ammonium carbamate.
8 er the conjugates previously connected via a carbamate.
9 to convert all primary amines to less basic carbamates.
10 reaction of N-arylhydroxylamines with diene carbamates.
11 )alkylboronates to enantioenriched lithiated carbamates.
12 HAS permit formation of chemically distinct carbamates.
13 ciations with, respectively, pyrethroids and carbamates.
14 ngement reactions of the corresponding allyl carbamates.
15 nt role in natural remediation mechanisms of carbamates.
16 ed secondary dialkyl TIB esters, but not the carbamates.
17 f alpha-lithiated haloalkanes, epoxides, and carbamates.
18 kinetically different for the two classes of carbamates.
19 n then be readily converted to carbonates or carbamates.
20 sing on the new class of N-(2-oxo-3-oxetanyl)carbamates.
21 tonated metal hydroxamates and lead to metal carbamates.
22 pyrethroids, and 1.5 (95% CI: 0.5, 4.8) for carbamates.
23 arbamates 5-7 (Scheme 2 ) and meta-protected carbamates 14, 15, and 20 (Schemes 5 and 7 ) by s-BuLi/(
24 methyl-N-[(2S,3R)-2-methyl-4-oxo-oxetan-3-yl]carbamate (14q) as the first single-digit nanomolar inhi
25 luorobenzoyllysineoxypentanedioic acid (OPA) carbamate [(18)F]23 and 4-iodo-2-[(18)F]fluorobenzoyllys
26 and 4-iodo-2-[(18)F]fluorobenzoyllysine OPA carbamate [(18)F]24 in particular exhibited high target-
28 rnal standard instead of less similar propyl carbamate; (2) extraction by diethyl ether instead of mo
30 l-carbamate (34) and 2-ethyl-3-methyl-pentyl-carbamate (38) also exhibited potent activity in the pil
33 r functionalized tertiary N,N-dialkyl aryl O-carbamates 5-7 (Scheme 2 ) and meta-protected carbamates
37 alkyl electrophile to generate a substituted carbamate, a process that has not been achieved effectiv
38 y of functional groups, such as an olefin, a carbamate, a thiophene, and a pyridine, and it has been
39 2,3-substituted-phenyl)piperazine-1-yl]alkyl]carbamates, a novel class of molecules that had shown pr
40 Two chemical probes, Azido Benzyl ferrocene carbamate (ABFC) and N-alkyl Azido Benzyl ferrocene carb
41 ligand paradigm was applied to the design of carbamates able to simultaneously target the recently pr
43 Above room temperature, both types of oxime carbamate acted as selective new precursors for aminyl a
49 e resulted in a soluble, orally bioavailable carbamate analogue providing identical activity in the a
51 les bearing both a lipophilic P2 isoindoline carbamate and a P1/P1' acylsulfonamide/acylsulfamide car
56 nitrogen nucleophiles such as sulphonamides, carbamates and amides have been shown to be appropriate
59 l adsorbs CO2 via formation of both ammonium carbamates and carbamic acid pairs, the latter of which
60 hroids, DDT and dieldrin, moderate level for carbamates and full susceptibility to organophosphates.
61 ross-coupling reaction of stereodefined enol carbamates and Grignard reagents to yield tri- and tetra
62 is strategy for the preparation of energetic carbamates and nitrocarbamates starting from readily ava
65 to the formation of the corresponding amine carbamates and protonated amines that were identified by
66 ity of two common protected forms of amines (carbamates and sulfonamides) to serve as directing group
69 mines, amides, isocyanates, isothiocyanates, carbamates and thiocarbamates with OH radicals within a
70 s based on labeled carboxylic acids, amides, carbamates and ureas now account for a substantial numbe
71 -ides to tert-butyl (S)-(3-oxopent-4-yn-2-yl)carbamate, and their structures were determined by NMR,
72 the OCH(2) linkage was replaced with amide, carbamate, and urea functionality, were investigated as
74 dissolving-metal cleavage of hindered phenyl carbamates, and an aminoiodocyclization to form the pyrr
76 f mesylates, sulfamates, esters, carbonates, carbamates, and methyl ethers as C-O-based electrophiles
78 , and imides (i.e., benzamides, tosylamides, carbamates, and phthalimide) to form the corresponding N
80 chemical methodologies for the synthesis of carbamates, and recent applications of carbamates in dru
82 of N-(2-(2-phenylthiazol-4-yl)ethyl)amides, carbamates, and ureas, which rapidly, selectively, and p
83 ative conjugate addition of a thiourea-bound carbamate anion to a vinyl phosphonium ion resulting fro
87 e with 6-aminoquinolyl-N-hydroxysuccinimidyl carbamate (AQC) for the determination of amino acids was
88 n with 6-aminoquinolyl-N-hydroxysuccinimidyl carbamate (AQC) in balsamic, apple, and red, white, and
89 N-Terminal Ser residues containing an Fmoc carbamate are converted into 2-(9'-fluorenylmethyloxy)-2
90 ates, including protonation constants of the carbamate, are reported for amines that follow this path
92 ibrium during the 4 h study period, suggests carbamates as alternative scaffolds for mitigating dose
93 ed variants of proline and the corresponding carbamate, as well as the four proline residues of an Sr
94 , carboxylic acids, amides, isocyanates, and carbamates, as well as tetrahydrofuran and gamma-butyrol
96 ectivity over hAChE was synthesized based on carbamates attached to tetrahydroquinazoline scaffolds w
97 two prodrug strategies, 1,4,2-dioxazole and carbamate, based on our 1-adamantylacetohydroxamic acid
100 d with 6-aminoquinolyl-N-hydroxysuccinimidyl carbamate before analysis using liquid chromatography el
103 methrin) insecticide in the first year and a carbamate (bendiocarb) insecticide in the two subsequent
104 Herein we demonstrate that N-acyl-tert-butyl-carbamates (Boc) and N-acyl-tosylamides (Ts), two classe
106 anes, sugar moieties, azetidines, tert-butyl carbamates (Boc-group), cyclobutanes, and spirocycles.
107 elatively quickly from the oil depot and its carbamate bond was too stable to be used as a prodrug.
108 primary and secondary amines via an amide or carbamate bond; however, the ability to employ tertiary-
109 dly release curcumin in vitro via degradable carbamate bonds, and retain in vitro bioactivity against
110 lling of Cx26 demonstrated that the proposed carbamate bridge between Lys125 and Arg104 biases the he
111 ly in the absence of a catalyst; the product carbamates can serve as useful intermediates in organic
112 th EPR and UV-vis spectroscopy indicate that carbamates can undergo direct reactions with various rad
116 ambda(6),2-benzothiazol-2- yl)methyl]benzoyl}carbamate CU-CPD103 (103), as a potent inhibitor using a
119 nt of the inhibitory potency of beta-lactone carbamate derivatives for NAAA and the identification of
120 nate, O-phenyl carbamate, urea, and N-phenyl carbamate derivatives of SB-3CT, a selective and potent
124 fied to ~0.58 mol, with ~0.15 mol in form of carbamate dianions and ~0.43 mol in form of carbamic aci
125 o-Diels-Alder reaction of nitrosoarenes with carbamate-dienes afforded cis-3,6-disubstituted dihydro-
128 ase biosensor was developed for detection of carbamate drugs based on TTF-TCNQ-ionic liquid gel thioc
130 9-xanthydrol for the determination of ethyl carbamate (EC) in wine by a previous high performance li
134 emonstrated that the use of nonracemic allyl carbamates enables the synthesis of enantioenriched benz
135 methylenedioxy, carbonate, cyclic carbonate, carbamate esters, and esters containing active transport
136 d cascade transformation involving a primary carbamate, ethyl glyoxylate, and various types of nucleo
137 not demonstrate cellular activity, however, carbamates exhibited cellular potency with the most acti
138 hyl N-(6-phenylsulfanyl-1H-benzimidazol-2-yl)carbamate) exhibits a potent growth-inhibitory activity
140 ed, encompassing an allyloxycarbonyl (Alloc) carbamate for Nalpha, a tert-butyl ester for the delta-C
142 d kinetic capture-and-release tests show the carbamate formation rate is fast enough to capture carbo
143 f the amines, that is CO(2) hydration and/or carbamate formation, is examined and, based on the mecha
144 urther synthetic manipulations involving the carbamate formation, lactone reduction and cyclization,
146 mate analogs, alpha-GalCer-6''-(pyridin-4-yl)carbamate, formed novel interactions with the NKTCR.
148 tethered aminohydroxylation of a homoallylic carbamate function and a Petasis Borono-Mannich addition
149 we demonstrate that neuroprotective aromatic carbamates function to increase the Bcl-2/Bax ratio to a
150 rimary and secondary amines to less reactive carbamate functional groups, indicated that primary and
152 udies in pancreatic cancer cells showed that carbamate functionalization of the 4-amino group of gemc
153 compounds (formaldehyde, acetaldehyde, ethyl carbamate, furan, furfural and acrolein) found in wines.
154 deoxy-D-galactopyranosylidene)amino N-phenyl carbamate (GalPUGNAc), N-acetyl-D-glucosamine-thiazoline
155 ition to alkenes, and cleavage of the methyl carbamate gives the free aminocyclopropanes as their HI
159 cular, hydrogen-bonding interactions through carbamate groups were found to be especially useful at d
161 sters) and secondary dialkyl N,N-diisopropyl carbamates have been reported to be resistant to deproto
163 and associated docetaxel hydroxy-tert-butyl carbamate (HDTX) metabolite biliary excretion, were best
164 ubstituents were used to control the rate of carbamate hydrolysis and the resulting protein release.
165 chemical groups: derivatives of (i) N-(tosyl)carbamate, (ii) p-toluenesulfonamide (PTSA), (iii) 4,4'-
166 ensation of the remaining ketone with methyl carbamate in the presence of acid initiated the programm
173 constants for the formation of carbamic acid/carbamates, including protonation constants of the carba
174 maticity of aromatic repeating units in poly(carbamates) increase the overall depolymerization rate.
175 get site loci (e.g. the Ace-1 target site of carbamate insecticides) or detoxification genes has been
177 mation of a putative alpha-chloro pyridinium carbamate intermediate, which appeared to readily underg
179 he tetrahydroquinazoline scaffold guides the carbamate into a close position to the active site.
180 transform di- and trisubstituted homoallylic carbamates into [4.1.0]-carbamate-tethered aziridines in
181 und n-alkylammonium oleate, phosphonate, and carbamate ion pairs that bind with greater affinity than
182 3 T) (13)C{(1)H} cross-polarization MAS NMR, carbamate is confirmed through splitting of the (13)C re
183 ecies that is either bicarbonate or a second carbamate is evident from bimodal T2 decay times of the
184 ecies in the near-surface region, while only carbamate is formed in the bulk, to differences in solva
185 a ring-closing metathesis reaction of allyl carbamates is presented as a method for the preparation
186 The epoxides, but not their urea, amide, or carbamate isosteres, impaired ATP production, enhanced c
189 analogue conjugated to the B12(2-) core via carbamate linkage and a fluorescein molecule attached at
190 ilic addition of free hydroxyl groups to the carbamate linkages and exhibits an Arrhenius activation
191 inating, electron-withdrawing benzyl alcohol-carbamate linker offers a probe having selective, sensit
192 factant containing an acryloyl amide tail, a carbamate linker, and a leucine headgroup of different c
194 elieve that tethering proteins by degradable carbamate linkers is a promising strategy to control the
199 thyl-N-ethyl or N-methyl-N-(4-methoxyphenyl) carbamate moieties at positions 4, 6, or 7 conferred bot
200 ween the reactivities of two closely related carbamate moieties, the N-ethoxycarbonyl and the N-pheno
202 ng aziridinium intermediates with a tethered carbamate moiety) to give oxazolidin-2-ones was initiall
203 substituents located ortho or meta to the O-carbamate moiety, and O-carbamate N-substituents was inv
206 aterials such as hydroxamic acids, N-hydroxy carbamates, N-hydroxyureas, nitrile oxides, and 1,2,4-ox
207 te (ABFC) and N-alkyl Azido Benzyl ferrocene carbamate (NABFC) composed of azide trigger group were d
208 ate an array of functional groups, including carbamate NH, halogen, nitrile, olefin, ketone, and este
209 port, we address the challenge of coupling a carbamate nucleophile with an unactivated secondary alky
210 allenyl and propargyl esters with N-methoxy carbamate nucleophiles to yield alpha,beta-unsaturated g
211 enantioenriched primary/secondary lithiated carbamates or benzoates to give 1,3-bis(boronic esters),
213 lectrostatic surface potential of a carbonyl/carbamate oxygen atom present in most KCNQ activators.
215 e, synthetic pyrethroid, organophosphate and carbamate pesticide residues in fruit juices using ultra
216 common organophosphorus, organochlorine and carbamate pesticides by 30-70% on tomato, rice, tea, bro
218 sy carbon electrode (GC), and used to detect carbamate pesticides in fruit and vegetables (apple, bro
226 age was attained by the glycosylation of 2-N-carbamate-protected alpha-GlcN-lactol with N-phenyl-trif
227 lladium-catalyzed ortho-arylation of diethyl carbamate-protected estrone and estriol with aryl iodide
228 des, dipeptides, and tripeptides whereas its carbamate-protected form adopts trans-conformation.
229 rmer specificity of delta-azaproline and its carbamate-protected form in linear and cyclic peptides w
230 sh studies with allyl, propargyl, and benzyl carbamate-protected rhodamines confirmed N-Poc as the mo
234 demonstrated, a rearrangement of (S,Z)-allyl carbamates provides (S)-teriary allylamines, whereas the
236 2-deoxy-D-glucopyranosylidene)amino N-phenyl carbamate (PUGNAc), O-(2-acetamido-2-deoxy-D-galactopyra
237 urotoxic pesticide groups (organophosphates, carbamates, pyrethroids, neonicotinoids, and manganese f
238 A variety of N-(1-methoxyalkyl)amides or carbamates react readily with sodium aryl sulfinates in
239 abeled with this reagent comprised of an NHS-carbamate reactive group, a quinoline fluorophore, and a
240 ve, we present properties and stabilities of carbamates, reagents and chemical methodologies for the
241 designed to be activated by hydrolysis of a carbamate releasing the free drug without the cleavage r
242 d method was optimized for the extraction of carbamate residues from a wide variety of fresh herbal p
245 o-4-((4-(trifluoromethyl)benzyl)amino)phenyl)carbamate (RL648_81), a new KCNQ2/3-specific activator t
246 e chemisorption reaction outcomes, including carbamate (RnNCOO(-)), carbamic acid (RnNCOOH), and bica
248 the CO2 carrier species, much the same as a carbamate serves as the CO2 carrier for amine-based capt
253 s use of alpha-lithio vinyl bromide or vinyl carbamate species, for which application to Zweifel-type
254 oposed mechanism involves protonation of the carbamate species, nucleophilic attack of the carbamic a
255 (-)-sparteine pair versus N,N-dialkyl aryl O-carbamate starting materials, temperature, solvents, ele
256 te terminal iron carbynes possessing an aryl carbamate substituent owing to the direct attachment of
257 ighly effective Diels-Alder reaction using a carbamate-substituted siloxy diene accompanied by a spon
259 reaction of the melampomagnolide-B-triazole carbamate synthon 6 with various terminal diamino- and d
260 stituted homoallylic carbamates into [4.1.0]-carbamate-tethered aziridines in good yields and with ee
261 design principles for creating aromatic poly(carbamates) that depolymerize from head-to-tail in low d
262 ure was observed including carbamic acid and carbamate, the former disappearing upon evacuation of th
266 The exposure to furan, acrolein and ethyl carbamate through wine consumption may pose risks to con
267 , largely because of their potential to form carbamates through H(2)N(delta(-))...C(delta(+))O(2) int
268 as electrochemically modified using ammonium carbamate to make it suitable for sensing free chlorine
273 AH covalent adducts, derived from the O-aryl carbamate URB597 and from the N-piperazinylurea JNJ16616
275 lti-dose intraperitoneal injections of ethyl carbamate (urethane, 1 g/kg body weight) were establishe
276 Hofmann rearrangement of carboxamides to carbamates using Oxone as an oxidant can be efficiently
281 rbents that uptake CO2 primarily as ammonium carbamates, we observe using solid state NMR that the ma
282 phophates, organochlorines, pyrethroids, and carbamates were aggregated within 1.25-km, 1.5-km, and 1
283 armacophores in place at C24, morpholines or carbamates were installed at the C3 position to refine t
287 of reaction products also shifts to ammonium carbamate when water vapor is present; a new finding tha
288 The CO2 adduct of 1,2-azaborine is a cyclic carbamate which undergoes photocleavage, thus resulting
289 (ca. twenty days) for quantification of five carbamates widely applied on tomato and potato crops.
292 e PIs incorporate various alcohol-derived P2 carbamates with acyclic and cyclic heteroatomic function
293 available olefins to internal vicinal fluoro carbamates with high regioselectivity (N vs F), many of
295 when applied to hindered systems (secondary carbamates with tBu-boronic esters) for the construction
296 constants for the formation of carbamic acid/carbamates with the protonation constant of the amine is
298 n achieve the coupling of a range of primary carbamates with unactivated secondary alkyl bromides at
299 opy, CO2 is found to be bound in the bulk as carbamate (with nominally 0.5 mol of CO2 bound per 1 mol
300 hosphate buffers) only 3% of 9-xanthyl ethyl carbamate (XEC) decomposes in approximately 48h, allowin
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