ライフサイエンスコーパス: inhibitory activity

1 CysC monomers and completely retain protease inhibitory activity.

2 tiestrogenic activity with the mitochondrial inhibitory activity.

3 imizing bioactive metabolites and tyrosinase inhibitory activity.

4 ical scavenging activities and LDL oxidation inhibitory activity.

5 that Dectin-3 is required for optimal growth-inhibitory activity.

6 athway signaling disruptor that lacked Hsp90 inhibitory activity.

7 between alpha-sheet structural stability and inhibitory activity.

8 ble for conferring alpha-sheet stability and inhibitory activity.

9 and selective Brr2 inhibitor 9 with helicase inhibitory activity.

10 for their antioxidant and alpha-glucosidase inhibitory activity.

11 N-benzylated derivative showed enhanced Clk1 inhibitory activity.

12 spho-mimetic mutation (T592E), abrogated the inhibitory activity.

13 t likely to yield derivatives with high Top1 inhibitory activity.

14 were synthesized and tested for 17beta-HSD14 inhibitory activity.

15 Y0123), and 47 (NY0173)) with low micromolar inhibitory activity.

16 f at least one phenyl ring is beneficial for inhibitory activity.

17 nding alone was not sufficient for ANGPTL4's inhibitory activity.

18 penetrate cells in culture, retaining HIV-1 inhibitory activity.

19 a-helix, accompanied by attenuation of NMDAR inhibitory activity.

20 n-MLL inhibitors considerably improved their inhibitory activity.

21 hment, as VLDL-depleted mouse serum lost HCV-inhibitory activity.

22 CB to wheat bread significantly increased XO-inhibitory activity.

23 closan may be related to their mitochondrial inhibitory activity.

24 agents exerting partial FXR agonism and sEH inhibitory activity.

25 mbinations with greater than additive growth-inhibitory activity.

26 nding may be the molecular mechanism for its inhibitory activity.

27 cancer cell lines and for protein synthesis inhibitory activity.

28 explains their extensive contribution to the inhibitory activity.

29 tor, or iniparib (n = 11), which has no PARP inhibitory activity.

30 ol content (GAE) and yeast alpha-glucosidase inhibitory activity.

31 predicted which genera were associated with inhibitory activity.

32 n and IC50 value of 1.60mg/ml for tyrosinase inhibitory activity.

33 es, revealing the structural basis for their inhibitory activity.

34 y test and only CSP4 and CSP6 exhibited high inhibitory activity.

35 her self-assembling abilities exhibit higher inhibitory activities.

36 cessed through ORAC, DPPH scavenging and ACE-inhibitory activities.

37 rates were assessed for their in vitro ACE-I inhibitory activities.

38 abolites were tested for NF-kappaB and K-Ras inhibitory activities.

39 lfonamide binding correlates well with their inhibitory activities.

40 ntibacterial, herbicidal, and various enzyme inhibitory activities.

41 t as well as superior antioxidant and enzyme inhibitory activities.

42 in vitro CB1R antagonist activities and iNOS inhibitory activities.

43 temperature, gave the highest alpha-amylase inhibitory activity (57.5%).

44 42.2%) and FRAP (0.81 mM)) and alpha-amylase inhibitory activity (62.1%), was then subjected to LCMS

45 Tyr-Pro had the highest ACE inhibitory activity (ACE IC50=5.21+/-0.94muM).

46 The compounds were tested for their inhibitory activities against BCRP and screened against

47 For the most promising compounds, the inhibitory activities against DNA gyrase from Staphyloco

48 zed molecule was generated with differential inhibitory activities against DprE1 and CYP2C9, which pr

49 opargylamines was synthesized and tested for inhibitory activities against monoamine oxidases.

50 (MIC50 = 1.56-6.25 mug/mL) and strong enzyme inhibitory activities against the bacterial phosphotrans

51 identified eight compounds with significant inhibitory activities against these proteins, two of whi

52 Rhp-PSP exhibited significant inhibitory activities against tobacco mosaic virus (TMV)

53 he new Top1 inhibitors also possess moderate inhibitory activities against tyrosyl-DNA phosphodiester

54 Comparisons of the enzyme inhibitory activity against a panel of HDAC isoforms rev

55 cetone extract of Undaria pinnatifida showed inhibitory activity against alpha-amylase, IC50 0.74+/-0

56 The tested T. terrestris and chickpea showed inhibitory activity against alpha-glucosidase (IC50 6967

57 o translates to a ~10-50-fold greater growth-inhibitory activity against breast cancer cell lines.

58 y activity against class IIa HDACs, but weak inhibitory activity against class I HDACs.

59 isoforms revealed these compounds had strong inhibitory activity against class IIa HDACs, but weak in

60 h carbon linkages had improved stability and inhibitory activity against FimH.

61 Phenolic compounds, their inhibitory activity against fungal amylase and the occur

62 )acetamide derivatives, showed low nanomolar inhibitory activity against hCA II and hCA VII, isoforms

63 -3503 and rac-cryptopleurine, exhibit potent inhibitory activity against hepatitis C virus (HCV) repl

64 Pleasingly, (IZ14N24N)3 possessed promising inhibitory activity against HIV-1 infection and markedly

65 emotype consistently conferred low nanomolar inhibitory activity against HIV-1.

66 ther, RGD-M/sPMI exerted potent tumor growth inhibitory activity against human glioblastoma in nude m

67 in the plant into two fragments, both having inhibitory activity against lignification.

68 ) using MTT assay, where they showed highest inhibitory activity against MCF-7.

69 E209 has potent nanomolar inhibitory activity against multiple strains of P. falci

70 amide derivatives (2 and 3) exhibited growth inhibitory activity against Mycobacterium tuberculosis (

71 oderate to weak cytotoxicity and significant inhibitory activity against nitric oxide (NO) production

72 DJK-5 showed stronger inhibitory activity against P. aeruginosa associated wit

73 zo[d]isothiazol-3(2H)-ones display nanomolar inhibitory activity against P. falciparum and P. vivax I

74 ed immunoglobulin G showed functional growth inhibitory activity against P. falciparum in vitro.

75 lead optimized NSC319726 and its reasonable inhibitory activity against pathogens suggest advancing

76 isplay reduced binding to LRP1 and unaltered inhibitory activity against prototypic metalloproteinase

77 ur compounds were further screened for their inhibitory activity against recombinant HDAC1-3, HDAC6,

78 ibitors were evaluated in screens for enzyme inhibitory activity against schistosome and human HDACs.

79 ime of 25 min, the hydrolysates demonstrated inhibitory activity against several gram-positive and gr

80 ain of the transcription factor STAT5 confer inhibitory activity against STAT3.

81 L7095) was also found to possess comparable inhibitory activity against T cells, indicating a potent

82 These compounds all displayed strong inhibitory activity against T.b. brucei but none of them

83 However, N-TIMP-3 displayed profound inhibitory activity against the D362H variants with a re

84 e flea, Xenopsylla cheopis, that exhibits an inhibitory activity against the NaV1.5 channel with an I

85 These antibodies exhibited a hierarchy of inhibitory activity against the NF54 laboratory strain o

86 ed aporphinoid alkaloids that exhibit potent inhibitory activity against the opportunistic fungal pat

87 drug, ELQ-334, demonstrated excellent growth inhibitory activity against the parasite, with potency e

88 ammary epithelial cells, possesses intrinsic inhibitory activity against triple-negative breast cance

89 anti-inflammatory properties and cell growth inhibitory activity against tumor cells.

90 es to elucidate the molecular basis of their inhibitory activities and an unconventional resistance m

91 The potent aromatase inhibitory activities and high ER-alpha and ER-beta bind

92 uents, resulting in compounds with high Top1 inhibitory activities and potent cytotoxicities in human

93 gest that HAX-1 is a major mediator of PLN's inhibitory activity and a critical gatekeeper of SR calc

94 roup gave analogue 7 with potent cell growth inhibitory activity and an activity profile similar to t

95 A-Top1 ternary cleavage complex, affect Top1 inhibitory activity and cytotoxicity.

96 protein co-precipitates showed improved ACE inhibitory activity and diminished antioxidant potency c

97 ied a set of compounds with the desired dual inhibitory activity and enhanced antiproliferative activ

98 protein co-precipitates showed decreased ACE inhibitory activity and increased antioxidant activities

99 milk of HIV-positive mothers has potent HIV-inhibitory activity and indicate that breast milk can pr

100 emical characteristics of milk's in vivo HIV-inhibitory activity and its ability to inhibit other mod

101 med by our research group have reported high inhibitory activity and potential agricultural and medic

102 PNN removal caused reduced inhibitory activity and reset the network to a juvenile

103 eptide aldehyde, which bears potent protease inhibitory activity and selectively targets a subset of

104 Quinoline-based analogues showed lower inhibitory activity and selectivity.

105 y profile allowing enhancement of proteasome-inhibitory activity and specificity of BTZ by endocytosi

106 The angiotensin I-converting enzyme (ACE) inhibitory activity and structural properties of oven-dr

107 positive correlation detected between their inhibitory activity and the reduction in cell migration.

108 ells (Bregs) enabling Tregs to recover their inhibitory activity, and in turn, leading to the rapid a

109 reased angiotensin I-converting enzyme (ACE) inhibitory activity, and in vitro gastrointestinal diges

110 GF WSP possessed NO inhibitory activity, and the strongest was GF121.

111 All inhibitory activities are dependent on three lysine resi

112 Their kinase inhibitory activities are mediated by a homologous N-ter

113 alpha-Conotoxin ImI displayed inhibitory activity as well.

114 ith histones was independent of its protease inhibitory activity, as demonstrated by the use of react

115 ses ChEMBL and PDB for fragments showing PDE inhibitory activity, as well as SureChEMBL for recent PD

116 nalysis of in vivo FLT3 inhibition by plasma inhibitory activity assay and indicated improved overall

117 tent human ether-a-go-go-related gene (hERG) inhibitory activity, associated with long Q-T syndrome,

118 benzyl-N-alkyloxy coumarins 2-12 showed good inhibitory activities at MAO-B, AChE, and BChE but low s

119 lues >10 mg/ml for a few or in most cases no inhibitory activity at all.

120 d the chalcone-derivative 8 possessing Notch inhibitory activity at low micro molar concentration in

121 ples showing more than 60% alpha-glucosidase inhibitory activity, at a concentration of 1 mg/ml, were

122 connectivity, leading to altered excitatory/inhibitory activity balance.

123 hese "hybrids" not only excel in outstanding inhibitory activity but also show high selectivity to PI

124 ar risk as NSAIDs with less cyclooxygenase-2 inhibitory activity, but at the cost of not controlling

125 u tail (IDL) that dramatically increased the inhibitory activity by up to 100 folds.

126 -precipitates showed increased alpha-amylase inhibitory activity compared to non-sonicated samples.

127 HG demonstrated the highest ACE-inhibitory activity, DPPH, ABTS radical scavenging activ

128 t a related compound lacking tyrosine kinase inhibitory activity, DV2-103, exerts similar effects on

129 cted its possible ligands and assessed their inhibitory activity experimentally.

130 ated strong antiflaviviral effects, and this inhibitory activity extended to other viruses, including

131 basophil activation and measurement of serum inhibitory activity for allergen-IgE binding to B cells

132 vailable antifolate with potent and specific inhibitory activity for aminoimidazole-4-carboxamide rib

133 The compounds showed practically no inhibitory activity for concentration of pyrrolidines in

134 his difference revealed a differential PARP3 inhibitory activity for each compound and a higher level

135 IgG4 including SIgE/IgG4 ratio), (iii) Serum inhibitory activity for IgE (IgE-FAB and IgE-BF), (iv) B

136 Serum inhibitory activity for IgE-FAB and basophil histamine r

137 bioactivities (ORAC, DPPH scavenging and ACE-inhibitory activities) generated from alkali extracted H

138 1.432mumol Trolox eq./mumol peptide) and ACE inhibitory activities (IC50=44-120muM).

139 entene core structure exhibits the strongest inhibitory activity (IC50 = 0.3-4.1 nM) against several

140 get hit compound (5b) exhibiting high hMAO B inhibitory activity (IC50 = 30 nM) and good MAO B/A sele

141 unds 1 (X80), 22, and 24 displayed excellent inhibitory activity (IC50 of 0.82 +/- 0.18 muM and 1.3 +

142 rimidine-2,4-diamine) that contribute to its inhibitory activity (IC50 value) and chaperoning efficac

143 subfraction, with enhanced alpha-glucosidase inhibitory activity (IC50=6.15mug/mL), with castalagin (

144 These quinolinol analogues demonstrated inhibitory activity in a cell-based model for SNAP-25 cl

145 nal in vitro assay to quantify their binding-inhibitory activity in a cohort of 466 rural Amazonians

146 Ag receptor ligation, we find that FCRL4 has inhibitory activity in cells coexpressing FGR but an act

147 ntibodies showed more potent parasite growth inhibitory activity in combination than on their own, su

148 Median Escherichia coli inhibitory activity in CVL specimens decreased significa

149 4 and 6 with preclinical evidence of growth-inhibitory activity in oestrogen receptor-positive breas

150 inal (BET) family proteins have shown growth-inhibitory activity in preclinical models of CRPC.

151 uation of antiproliferative effects and HDAC inhibitory activity in the human ovarian cancer cell lin

152 Imbalance between excitatory and inhibitory activity in the LH can induce changes in food

153 ng memory load and the balance of excitatory/inhibitory activity in the motor cortex and potentially

154 Best inhibitory activity (in the low nanomolar-subnanomolar r

155 aR isomers of 1 had a critical effect on the inhibitory activity, indicating that modulation of the c

156 elective, and reversible monoamine oxidase B inhibitory activity is a clinically relevant subject.

157 The ability of EGCG to mediate its inhibitory activity is counter-regulated by the presence

158 t not to the LAP isoform, explaining why its inhibitory activity is selective for LAP*.

159 ntioxidant properties, strong cholinesterase inhibitory activity, less hepatotoxicity than tacrine, a

160 f Kh1 and En samples showed moderate to good inhibitory activities (MICs=62.5-125mug/ml) against thre

161 igh-throughput screening was used to measure inhibitory activities of BKIs against C. parvum in vitro

162 The chemotaxis inhibitory activities of both compounds were confirmed i

163 stant region dramatically enhanced the tumor inhibitory activities of KTN0073 but not KTN0074, sugges

164 The inhibitory activities of T. terrestris and chickpea agai

165 The antioxidant and ACE-inhibitory activities of the extracted proteins were ini

166 sEH inhibitory activity of (18)F-FNDP was measured using an

167 e (1 mg/ml), that demonstrated highest ACE-I inhibitory activity of 70.37%, was characterised in term

168 Here, we report the inhibitory activity of a flavone rich extract "430D-F5"

169 iation of an auxiliary domain stimulates the inhibitory activity of a Kunitz-type inhibitor (i.e. the

170 interplay between tertiary structure and the inhibitory activity of a multidomain protease inhibitor.

171 LC-HRMS-SPE-NMR showed the alpha-glucosidase inhibitory activity of A. nodosum, F. vesoculosus, Lamin

172 , these findings pave the way to explore the inhibitory activity of Amt-related analogues in mutated

173 n interactions have evolved to stimulate the inhibitory activity of an integrated Kunitz.

174 The biofilm-inhibitory activity of antibiotics and/or the anti-biofi

175 he absence of vivax invasion assays, binding-inhibitory activity of antibodies has been reported to b

176 escribed herein possess the most potent CD38 inhibitory activity of any small molecules described in

177 The trypsin inhibitory activity of BG-4 is 8.6 times higher than pur

178 The high trypsin inhibitory activity of BG-4 may be responsible for its c

179 ction of HVR1 antibodies should increase the inhibitory activity of broadly neutralizing anti-HCV ant

180 ion.IMPORTANCE The greater ex vivo antiviral inhibitory activity of CD8(+) T cells from elite control

181 In vitro assays revealed an inhibitory activity of coumaroylagmatine on P. infestans

182 which blocks Wnt secretion, enhances growth inhibitory activity of Erlotinib.

183 The cyclooxygenase enzyme inhibitory activity of extract and isolates at 100 mug/m

184 ely affected angiotensin I-converting enzyme inhibitory activity of fermented lentil (p<.0001).

185 separating the FLD from the CCD-mediated LPL-inhibitory activity of full-length Angptl4 reveals lipol

186 enolic composition and xanthine oxidase (XO) inhibitory activity of green coffee beans (GCB) and whol

187 een of a series of metal salts showed marked inhibitory activity of group 11 and 12 metals against th

188 of this study was to evaluate the potential inhibitory activity of guarana extracts, after digestion

189 The ACE-inhibitory activity of HG showed the highest stability a

190 Inhibitory activity of HNPs depends on the RRY motif tha

191 To test the newly discovered B cell-inhibitory activity of HSCs in vivo, we developed a prot

192 This direct B cell-inhibitory activity of HSCs should contribute to the mec

193 Highest ACE-inhibitory activity of hydrolyzed protein fractions was

194 The inhibitory activity of individual ISGs varies depending

195 Inhibitory activity of K12 was examined in vivo using a

196 f the internal domain but also stimulate the inhibitory activity of Kunitz-1.

197 Thus, the inhibitory activity of L-cIDPR analogues appears to depe

198 gulation appears to be the foundation of the inhibitory activity of many of the commercial herbicides

199 Herein, we present the synthesis and the inhibitory activity of novel and highly effective organo

200 We leveraged the powerful growth inhibitory activity of Nutlin-3a to select p53-mutated c

201 The ACE-inhibitory activity of OD-FPH was more stable (during se

202 ate that R292K, E119V, and I222K reduced the inhibitory activity of oseltamivir, not only in the NI a

203 ieves CDK2 inhibition by suppressing the CDK inhibitory activity of p27.

204 g that these regions are responsible for the inhibitory activity of PEX9.

205 e that this trapping mechanism underlies the inhibitory activity of potent M2 channel blockers, as su

206 zyme inhibition kinetics for calculating the inhibitory activity of protein anti-glycation agents.

207 The study suggested that the ACE inhibitory activity of protein hydrolysate was not affec

208 The angiotensin I-converting enzyme (ACE) inhibitory activity of protein hydrolysates from tilapia

209 nd the importance of membrane binding on the inhibitory activity of ProTx-II remain unknown.

210 alpha-helix most drastically suppressed the inhibitory activity of RD3 and disrupted RD3 co-localiza

211 zymes, consistent with a hypothesis that the inhibitory activity of RD3 has a functional role in phot

212 capacity and carbohydrate-hydrolysing enzyme inhibitory activity of roselle beverages during storage.

213 This inhibitory activity of RVB2 is antagonized by Env throug

214 Interestingly, unlike wild-type SBV, the inhibitory activity of SBVDeltaNoLS toward RNA Pol II tr

215 nfectivity, being required to antagonize the inhibitory activity of Serine incorporator (SERINC) prot

216 reticulocyte-binding properties and binding-inhibitory activity of specific anti-PvRBP2c/PvRBP1a hum

217 These two domains are required for the inhibitory activity of tau on EB localization to microtu

218 The latter blocks the inhibitory activity of the autoinhibitor domain.

219 The in vitro ACE inhibitory activity of the BSG-PI increased significantl

220 The inhibitory activity of the compounds against norovirus 3

221 tioxidant capacity and the alpha-glucosidase inhibitory activity of the duodenal extract correlated w

222 Here the synthesis and potent inhibitory activity of the first CYP26A1 selective inhib

223 reported structural assignment and elastase inhibitory activity of the isolated natural product were

224 o gastrointestinal digestion reduced the ACE inhibitory activity of the M hydrolysate but enhanced it

225 The inhibitory activity of the non-digested and digested sam

226 n correlated with transmission risk, the HIV-inhibitory activity of their breast milk has not been co

227 mportant interactions that contribute to the inhibitory activity of these compounds, and provide info

228 The species-selective inhibitory activity of these small molecules against Pla

229 The inhibitory activity of two compounds (51, 52) is compara

230 M domain, surprisingly, does not abolish the inhibitory activity of viperin against FPPS; indeed, som

231 enesis at the detriment of myogenesis and an inhibitory activity on angiogenesis.

232 w much endogenous HAX-1 contributes to PLN's inhibitory activity on calcium cycling is unknown.

233 s a result, these compounds also show growth inhibitory activity on cancer cells.

234 creases p27 levels, it also attenuates p27's inhibitory activity on CDK2 and thereby contributes to i

235 This compound was devoid of inhibitory activity on COX isozymes and blocked AKR1C3 m

236 We also show that the NS4 inhibitory activity on gene expression is related to its

237 nder certain circumstances, it also shows an inhibitory activity on metastatic processes, and the cau

238 ed comparable antioxidant capacity, stronger inhibitory activity on pancreatic lipase and comparable

239 dissociates it from 5'UTRs and relieves its inhibitory activity on RP mRNA translation.

240 Consistent with its inhibitory activity on the IRE1alpha-XBP1 branch of the

241 tor approved for the treatment of MF, had no inhibitory activity on this pathway.

242 Using agents that lack either RPE65 inhibitory activity or the capacity to sequester atRAL,

243 The pCQ also demonstrates superior inhibitory activity over HCQ when tested in a mouse mode

244 The alpha-amylase inhibitory activities ranged from 52.5 to 67.2mug/mL in

245 ng fermentation, while the alpha-glucosidase inhibitory activities ranged from 95.2 to 196.1mug/mL.

246 nt and angiotensin I converting enzyme (ACE) inhibitory activities released from lentil proteins by S

247 ip between ternary complex reversibility and inhibitory activities reported with cultured cells.

248 t effect and angiotensin I-converting enzyme inhibitory activity), rheological, and water mobility by

249 cyano and methoxy moieties with interesting inhibitory activity/selectivity against the tumor associ

250 A biochemical assessment of the inhibitory activity suggested that the S. caprae autoind

251 LRV1 lacks cis- or trans-acting RNAi inhibitory activities, suggesting that virus retention m

252 e synthase (iNOS) and cyclooxygenase (COX-2) inhibitory activity than an equivalent mixture of flavon

253 and pepsin hydrolysates exhibited higher ACE-inhibitory activity than HT (P<0.05).

254 orylated D-tetrapeptides exhibit more potent inhibitory activity than the diphosphorylated D-tetrapep

255 y such lipids, we pursued a Hedgehog pathway inhibitory activity that is particularly abundant in fla

256 nity than wild-type HVEM and retained potent inhibitory activity that reduced T-cell receptor, B-cell

257 ical inhibitors, we predicted their putative inhibitory activities to trypsin/chymotrypsin/elastase-l

258 no, nitro, acetamido, and fluoro led to high inhibitory activities toward ABCG2.

259 Investigations of the inhibitory activity toward ABCB1 and ABCC1 yielded a hig

260 esized compounds showed significantly higher inhibitory activity toward BChE with IC50 values in subm

261 Mac-1 exhibits a unique inhibitory activity toward IL-13-induced JAK/STAT activa

262 Besides the preservation of the TA inhibitory activity toward L. monocytogenes, the possibi

263 A structural analog of HS38, with inhibitory activity toward proviral integrations of Molo

264 combinant KT inhibitor (rFhKT1) exhibited no inhibitory activity toward serine proteases but was a po

265 le-3-carboxamide 8a, were found to show high inhibitory activity toward susceptible M. tuberculosis s

266 othelial progenitor EP cells) and the kinase inhibitory activity (toward both isolated kinases and EP

267 osed of Az and geldanamycin, which have high inhibitory activities towards both Hsp70 and Hsp90, exhi

268 wever, the Az and imatinib hybrids have weak inhibitory activities towards Hsp70 and Abl, and display

269 Novel indole derivatives with inhibitory activity towards acetyl/butyrylcholinesterase

270 stance to gastrointestinal digestion and the inhibitory activity towards endothelial cell migration.

271 (USP14) in vitro, with comparatively weaker inhibitory activity towards UCHL5 (ubiquitin-C-terminal

272 etection and quantification of alpha-amylase inhibitory activity using the glucose assay kit was deve

273 The range of the values for alpha-amylase inhibitory activity was 10.03-23.33mM, whereas the value

274 Interspecies conservation of this inhibitory activity was confirmed on TLR7/8 activity in

275 The inhibitory activity was determined using BAT inhibition

276 The PARP-1 inhibitory activity was evaluated for compound (1) (IC50

277 eparations of plant extracts, a strong TRPC6-inhibitory activity was found in conifer balsams.

278 The highest DPP-IV inhibitory activity was found with the amino acid Tyr (D

279 Higher ACE-inhibitory activity was generated in the trypsin and pep

280 activity whereas a negative impact on lipase inhibitory activity was observed (p<.0001).

281 t relationship between SCCD pressure and ACE inhibitory activity was observed, with 34.63, 38.75, and

282 Without PNNs, inhibitory activity was reduced, whereas spiking variabi

283 es to bind directly to PfHsp90 with their Pf-inhibitory activity, we found that these types of compou

284 reatment of R36A with trypsin eliminated its inhibitory activity, we incubated R36A in choline chlori

285 dant and angiotensin-converting-enzyme (ACE) inhibitory activities were measured.

286 lase and angiotensin converting enzyme (ACE) inhibitory activities were successfully identified using

287 as 10.03-23.33mM, whereas the values for ACE inhibitory activity were of 1.52-31.88muM.

288 lar dried Jameed also led to the highest ACE inhibitory activities whereas antioxidant activity was l

289 rolysates with potential antioxidant and ACE inhibitory activities, which can be used to obtain new a

290 ually dependent equilibria abrogated DB270's inhibitory activity, which was substantively restored un

291 N-FIV (3-1kDa) fractions showed the best ACE-inhibitory activities with IC50 values of 53.31 and 75.0

292 3a and 7c exhibited promising inhibitory activities with MICs ranging 1-8 mug/mL again

293 f synthesized 1 revealed increasing APOBEC3G inhibitory activity with age, suggesting that 1 decompos

294 The first peptide displayed the highest ACE inhibitory activity with an IC50 of 5.22muM.

295 void of antifungal and human cytochrome P450 inhibitory activity with excellent pharmacokinetics, saf

296 er-Val and Ile-Phe were shown to exhibit ACE inhibitory activity with IC50 values of 60.68+/-1.06 and

297 highest alpha-glucosidase and alpha-amylase inhibitory activity with IC50=1.1+/-0.1mug/ml and IC50=1

298 ed concentration-dependent alpha-glucosidase inhibitory activity with IC50=35.01 mug/ml.

299 r data demonstrate that RT53 possesses tumor-inhibitory activity with no toxicity in mice, suggesting

300 e of hydrolysis (DH)) showed the highest ACE inhibitory activity, with an IC50 value of 0.54mg/ml, wh