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1 LXRbeta agonism robustly suppressed tumor growth and met
2 LXRbeta gene expression poorly correlates with ABCA1 in
3 LXRbeta selectivity was confirmed using macrophages deri
4 LXRbeta subsequently modulates signaling by ALK-1 and th
5 LXRbeta targeting significantly prolonged animal surviva
6 LXRbeta was insensitive to fatty acid regulation in both
7 LXRbeta(-/-) mice responded to 24-h dehydration with a d
8 LXRbeta-deficient mice crossed to the hyperlipidemic Apo
12 ti-inflammatory activities and, in addition, LXRbeta is involved in the genesis of dopaminergic neuro
13 R modulator GSK9772 ( 20) as a high-affinity LXRbeta ligand (IC 50 = 30 nM) that shows separation of
14 ll agonist selectively kills GBM cells in an LXRbeta- and cholesterol-dependent fashion, causing tumo
15 l receptors LXR (liver X receptor)-alpha and LXRbeta are nuclear receptors that play a key role in re
20 of cofactor peptides onto both LXRalpha and LXRbeta and showed an EC(50) of approximately 2 muM in p
21 here that the nuclear receptors LXRalpha and LXRbeta and their oxysterol ligands are key regulators o
22 eceptors liver X receptor (LXR) LXRalpha and LXRbeta are differentially expressed ligand-activated tr
24 istochemical staining that both LXRalpha and LXRbeta are expressed in the cell nuclei of the epitheli
25 demonstrate here that although LXRalpha and LXRbeta are not required for adipocyte development per s
26 confirmed that 4 binds to both LXRalpha and LXRbeta directly and recruits coactivator peptide SRC-1.
27 derived from mice lacking both LXRalpha and LXRbeta failed to up-regulate the expression of ABC8 fol
28 addressed how deletion of both LXRalpha and LXRbeta from mouse liver (LXR double knockout [DKO]) aff
31 of the liver X receptors (LXRs) LXRalpha and LXRbeta in carbohydrate sensing by the liver (see the re
32 confirm an equivalent role for LXRalpha and LXRbeta in the regulation of ABCA1 and SREBP-1c gene exp
33 Desmosterol bound to purified LXRalpha and LXRbeta in vitro and supported the recruitment of steroi
34 at the liver X receptors (LXRs) LXRalpha and LXRbeta inhibit basal and cytokine-inducible expression
36 h deep sequencing revealed that LXRalpha and LXRbeta occupy both overlapping and exclusive genomic re
37 UMOylation of nuclear receptors LXRalpha and LXRbeta plays a critical role in the transrepression of
41 receptor coactivator-1 to human LXRalpha and LXRbeta with EC(50)s of 40 nM, profiles as an LXR agonis
43 ver X receptors alpha and beta (LXRalpha and LXRbeta) are important regulators of cholesterol homeost
45 ver X receptors alpha and beta (LXRalpha and LXRbeta) are oxysterol-activated transcription factors t
46 entified the liver X receptors (LXRalpha and LXRbeta) as important regulators of cholesterol and lipi
47 role of the liver X receptors (LXRalpha and LXRbeta) in preventing accumulation of free cholesterol
48 red that the Liver-X-Receptors (LXRalpha and LXRbeta), nuclear receptors known to regulate lipid meta
49 iver X receptors alpha and beta(LXRalpha and LXRbeta), which are important in regulating not only lip
51 is lost in animals lacking both LXRalpha and LXRbeta, confirming the critical role of these receptors
52 oxidized lipids, which activate LXRalpha and LXRbeta, resulting in the induction of ABCA1, ABCG1, and
57 eptors liver X receptor alpha (LXRalpha) and LXRbeta function as physiological receptors for oxidized
58 iver X receptor alpha (LXRalpha) (NR1H3) and LXRbeta (NR1H2) are important regulators of genes involv
59 ear oxysterol receptors LXRalpha (NR1H3) and LXRbeta (NR1H2) coordinately regulate the expression of
60 The liver X receptors, LXRalpha (NR1H3) and LXRbeta (NR1H2), are ligand-activated transcription fact
66 the same degree of potency as 22R-HC (3) at LXRbeta, while it was virtually inactive at LXRalpha (EC
68 lear receptor family, liver X receptor beta (LXRbeta) and thyroid hormone receptor alpha (TRalpha), h
70 udies have implicated liver X receptor beta (LXRbeta) in key neurodevelopmental processes and neurode
71 he oxysterol receptor liver X receptor beta (LXRbeta) in the etiology of diabetes insipidus (DI).
73 creased expression of liver X receptor beta (LXRbeta), a nuclear receptor that controls cellular lipi
74 the nuclear receptor, liver X receptor beta (LXRbeta), had an adverse effect on progression of the di
75 ncrease and activates liver X receptor beta (LXRbeta), promoting cholesterol release from lysosomes a
77 athway activation in macrophages achieved by LXRbeta and endogenous ligand is unable to maintain home
78 nts revealed these effects to be mediated by LXRbeta, which elicits these outcomes through transcript
79 female mice, we found that LXRs, especially LXRbeta, also repress the browning process of subcutaneo
80 ated transcriptional responses, establishing LXRbeta as a potential modulator/mediator of ALK-1/ALK-2
83 lude that the anxiogenic phenotype in female LXRbeta(-/-) mice is caused by reduced GABAergic input f
85 ompounds displayed good binding affinity for LXRbeta and LXRalpha and were potent activators in LBD t
86 Compound 13 demonstrated partial agonism for LXRbeta in kidney HEK-293 cells but did not activate Gal
90 skin, we mapped its cistrome by identifying LXRbeta-RXRalpha binding sites using ChIP-on-chip in nor
93 imilar food intake and oxygen consumption in LXRbeta-/- mice suggests that reduced storage of lipid i
94 dition, 22ROH did not reduce inflammation in LXRbeta-/- or LXRalphabeta-/- animals, indicating that L
95 nserved lysine (K432 in LXRalpha and K433 in LXRbeta) adjacent to the ligand-regulated activation dom
97 retarded migration of later-born neurons in LXRbeta(-/-) mice but that as thyroid hormone (TH) incre
101 the two isoforms of Liver X receptor (LXR), LXRbeta has been shown to have major effects in the cent
106 es from the livers of wild-type and LXRalpha/LXRbeta-null mice after exposure to the LXR agonist N-(2
107 r receptors, the liver X receptors (LXRalpha/LXRbeta), protects against atherosclerosis by transcript
109 heral tissues from these LXRalpha-null mice, LXRbeta activation increases ABCA1 and SREBP-1c gene exp
110 al docking studies using GLIDE with modified LXRbeta ligand-binding domain (LBD) on internal compound
113 XR activation promoted the direct binding of LXRbeta to the ligand-binding domain of ERalpha and init
115 normalities were detectable in the cortex of LXRbeta(-/-) mice and ApoER2 expression was much stronge
119 Cells with CRISPR-mediated knockdown of LXRbeta, but not ABCA1, had decreased cell cycle progres
123 aminergic neurons of the substantia nigra of LXRbeta(-/-) mice were much more severely affected by MP
129 activated ALK-1 results in translocation of LXRbeta from the nuclear compartment to the cytoplasmic
130 del of PD to investigate the possible use of LXRbeta as a target for prevention or treatment of PD.
136 ble, highly brain-penetrant LXRalpha-partial/LXRbeta-full agonist selectively kills GBM cells in an L
137 nuclear receptors, some of which (PPARalpha, LXRbeta) regulate specific liver gene expression network
139 t required for adipocyte development per se, LXRbeta is required for the increase in adipocyte size t
141 e that it is possible to achieve significant LXRbeta selectivity in a small molecule while maintainin
146 endothelial cells (ECs) and discovered that LXRbeta has nonnuclear function and stimulates EC migrat
147 optic nerve, providing in vivo evidence that LXRbeta deletion delays both oligodendrocyte differentia
148 or LXRalphabeta-/- animals, indicating that LXRbeta is required for this anti-inflammatory effect.
150 and lipidomics analyses cells revealed that LXRbeta regulates the expression of immune response gene
151 alysis of islet gene expression reveals that LXRbeta is required for expression of the cholesterol tr
152 Collectively, these results suggest that LXRbeta, by driving RGCs to become OPCs in the dorsal co
153 ncrease in urine osmolality, suggesting that LXRbeta is a key receptor in controlling water balance w
156 in NHEKs, demonstrating that 77% of all the LXRbeta-RXRalpha binding regions show the presence of AP
158 NS phenotype is much more severe than in the LXRbeta ko mice, suggesting a contribution of LXRalpha i
159 The reason for the migration defect in the LXRbeta(-/-) mouse and the possibility that TRalpha may
160 A comparison with existing structures of the LXRbeta homodimer and LXRalpha:RXR (retinoid X receptor)
162 Despite reduced amounts of adipose tissue, LXRbeta-/- mice on a chow diet have insulin sensitivity
163 lthough 13 showed potent binding affinity to LXRbeta (IC(50) = 53 nM), it had little binding affinity
168 the structurally related analog 19 bound to LXRbeta reveals regions within the receptor that can aff
172 The interaction of activated ALK-1 with LXRbeta in the cytoplasmic compartment results in the sp