ライフサイエンスコーパス: boronic acid

1 MR study of the protodeboronation of an aryl boronic acid.

2 on-promoted transmetalation reaction of aryl boronic acid.

3 which undergoes cross-coupling with the aryl boronic acid.

4 subtly changing the structure of the achiral boronic acid.

5 tected using the fluorescent probe, coumarin boronic acid.

6 ly handled and widely commercially available boronic acids.

7 of sulfur dioxide into (het)aryl and alkenyl boronic acids.

8 aryl phosphonium salts and coupled with aryl boronic acids.

9 sceptible to potent reversible inhibition by boronic acids.

10 anocatalytic strategy for the formylation of boronic acids.

11 dentifying bortezomib and additional peptide boronic acids.

12 ve coupling of methylene C-H bonds with aryl boronic acids.

13 y accessible from the commercially available boronic acids.

14 henols and naphthols using readily available boronic acids.

15 s, as well as arylammonium salts directly to boronic acids.

16 ing reaction of diaryl diselenides with aryl boronic acids.

17 les the generation of a variety of protected boronic acids.

18 al groups such as alcohols, amines, and even boronic acids.

19 clotrimers, which are readily intercepted by boronic acids.

20 ate for the reaction mechanism in Wulff-type boronic acids.

21 racemic fused bicyclic allylic chlorides and boronic acids.

22 des together with a variety of alkyl or aryl boronic acids.

23 ion followed by cross-coupling reaction with boronic acids.

24 lladium intermediate using 1.5 equiv of aryl boronic acid 2.

25 llowed by covalent coupling of 3-aminophenyl boronic acid (3-APBA).

26 rotocol provide details for preparation of a boronic acid (3-cyanopheylboronic acid) and a boronic es

27 alogue of the sensor that does not contain a boronic acid (4) responded nearly identically to 3 in th

28 Boronic acids act as Bronsted acid type receptors throug

29 A detailed investigation supports that boronic acid activation proceeds through hydrogen-bondin

30 shared the same functional groups (halides, boronic acids, alkenes, and alkynes, among other groups)

31 and Suzuki-Miyaura cross-coupling with aryl boronic acids allowed the synthesis of alpha-amino acids

32 omplexation of particular diol groups by the boronic acid also enables selective transformations of m

33 etrahedral adducts with the B(III) center of boronic acids, although there is also evidence for some

34 as solved through the development of a novel boronic acid-amine copromoter system for glycosyl accept

35 ming Petasis reaction occurring between aryl boronic acids, amines, and glyoxylic acids to prepare al

36 was used to attach the well-known anthracene-boronic acid (An-BA) probe to a biomimetic DNA scaffold

37 werful multicomponent coupling reaction of a boronic acid, an amine, and a carbonyl derivative.

38 Using a combination of boronic acid and 5-chlorosalicylic acid as the additives

39 Screening 3872 possible combinations from 44 boronic acid and 88 diol derivatives revealed several co

40 alysis indicated the association behavior of boronic acid and AHB.

41 Reaction occurring between boronic acid and cis-diol moiety of MAGs blocked the for

42 Boronic acid and esters have been extensively utilized f

43 d antibody immobilization via interaction of boronic acid and oligosaccharide moiety found on Fc regi

44 loyed readily available and benchmark stable boronic acid and potassium aryltrifluoroborate derivativ

45 via forming the cis-diol linkage between the boronic acid and sugar moieties.

46 Two additional processes compete when the boronic acid and the boronate are present in sufficient

47 pi interaction between the substrate ligated boronic acid and the phosphate.

48 means of electro-polymerization of 3-Thienyl boronic acid and Thiophen.

49 a stereodynamic probe carrying complementary boronic acid and urea units achieves this goal with hydr

50 ntional oxidative Heck reaction between aryl boronic acids and alkenes typically involved the Pd(II)/

51 ing reaction between readily available vinyl boronic acids and alkynes to provide unsymmetrical 3-bor

52 xpand this approach from the condensation of boronic acids and catechols to the dehydrative trimeriza

53 Coupling of readily available boronic acids and diazo compounds has emerged recently a

54 bioorthogonal click reaction between abiotic boronic acids and diols.

55 e reaction was amenable to a variety of aryl boronic acids and disubstituted malononitriles, providin

56 Aryl boronic acids and esters are important building blocks i

57 Boronic acids and esters have critical roles in the area

58 The widespread use of alkyl boronic acids and esters is frequently hampered by the c

59 Alkyl boronic acids and esters play an important role in the s

60 Many of the current applications of boronic acids and esters require materials with very low

61 ium catalyzed oxidative homocoupling of aryl boronic acids and esters to biphenyls has been recognize

62 thod of conversion of haloarenes directly to boronic acids and esters.

63 of the methylamino group to (hetero)aromatic boronic acids and esters.

64 rylating carbocyclization of allenynes using boronic acids and focuses on the correlation between rea

65 he coupling of aryl, heteroaryl, and alkenyl boronic acids and gives access to functionalized bicycli

66 y alkylboronate, and the preparation of free boronic acids and hemiboronic heterocycles.

67 ate to good yields via the reactions of aryl boronic acids and ortho-hydroxyarylaldehydes in the pres

68 rboxylates with vicinal donor aryl groups by boronic acids and potassium organotrifluoroborates under

69 vast reagent space of commercially available boronic acids and proceeds at ambient temperature.

70 cross a broad library of aryl and heteroaryl boronic acids and provides improved access to a fluoroge

71 Enantioconvergent arylation reactions of boronic acids and racemic beta-stereogenic alpha-keto es

72 ion and nitrosation) that involve the use of boronic acids and some of their derivatives as carbon-nu

73 originate from the stabilization of the (E)-boronic acids and the destabilization of the (E)-boronic

74 ) by a palladium-catalyzed cross-coupling of boronic acids and the thioimidate KAT transfer reagent.

75 Boronic acids and their derivatives are some of the most

76 These SCCs@MOFs catalyze the coupling of boronic acids and/or alkynes, representative multi-site

77 C-H bond (that is, a nitro group, halogen or boronic acid) and a subsequent functionalization or cros

78 mponent reaction involving terminal alkynes, boronic acids, and perfluoroalkyl iodides is presented h

79 phenols, diols, silanols, carboxylic acids, boronic acids, and phosphoric acids, were examined with

80 reacting flow-generated diazo compounds with boronic acids, and their application in controlled itera

81 Treatment of the 1,8-naphthalenediyl-bridged boronic acid anhydride 1 with LiAlH(4)/Me(3)SiCl afforde

82 co-functionalizing AuNPs with 3-aminophenyl boronic acid (APB) and L-glutamic acid-(2,2,2)-trichloro

83 Fluorinated boronic acid-appended benzyl bipyridinium salts, derived

84 We have prepared a new class of boronic acid-appended naphthyl-pyridinium receptor compo

85 strategy, we present the use of fluorinated boronic acid-appended pyridinium salts in combination wi

86 mponent probes were assembled with up to six boronic acid-appended viologens (BBVs): 4,4'-o-BBV, 3,3'

87 rs other than the Lewis acidity (pKa) of the boronic acid are at play.

88 Boronic acids are a well-known class of reagents that ha

89 ium catalyzed cross-coupling reactions using boronic acids are applied to aromatic and allenic compou

90 Boronic acids are centrally important functional motifs

91 Although boronic acids are recognized primarily for their utility

92 We show that pyridine boronic acids are unsuitable, but they can be halogen-mo

93 nd amines via (2-(thiophen-2-ylmethyl)phenyl)boronic acid as a highly active bench-stable catalyst.

94 Correction for 'Boronic acids as building blocks for the construction of

95 ic significance of this approach, with alkyl boronic acids as linchpins, is demonstrated through vari

96 e core have used organoboron dichlorides and boronic acids as the boron precursors.

97 The results can inform the use of boronic acids as they are increasingly utilized in the d

98 d-AAA) of acyclic alpha-hydroxyketones using boronic acids as traceless templates.

99 fluorination of allylic alcohols using aryl boronic acids as transient directing groups.

100 howed a good substrate scope with respect to boronic acids as well as 2-carbonyl-3-propargyl indoles

101 with a range of unactivated secondary Csp(3) boronic acids, as well as the stereocontrolled synthesis

102 time, a general, electrophilic amination of boronic acids at ambient temperature.

103 assisted amidation of readily available aryl boronic acids at room-temperature under open-flask condi

104 tidine residues direct oxidative coupling of boronic acids at the backbone NH of a neighboring amino

105 one can locally control the condensation of boronic acids at the liquid/solid interface.

106 study is reported where folic acid (FA) and boronic acid (BA) based cytosensors and their analytical

107 A multiligand set of boronic acid (BA) beta-lactamase inhibitors was obtained

108 phene nanoribbons (MGNRs) were modified with boronic acid (BA) to create a supporting matrix that is

109 l-known dynamic covalent interaction between boronic acids (BAs) and catechols (CAs) into synthetic n

110 able sensor is constructed of a fluorescent, boronic-acid based glucose indicating polymer coated ont

111 ts or through introduction of stoichiometric boronic acid-based additives.

112 study illustrates an approach for designing boronic acid-based chemoreceptors for the recognition an

113 at include antibodies, lectins, aptamers and boronic acid-based entities.

114 Using a well-known boronic acid-based saccharide sensor (3), this work reve

115 A magnetic graphene nanoribbon-boronic-acid-based immunosensor was developed and tested

116 as been designed such that the reaction with boronic acid bearing drugs induces an in situ self-assem

117 eficient, electron-rich or ortho-substituted boronic acids better results are obtained with racemic a

118 1,3-syn diol motifs showed high affinity for boronic acid binding.

119 )F singlets was utilized to characterize the boronic acid/boronate equilibrium kinetics.

120 s in the protic-solvent-inserted form of the boronic acid/boronate ester.

121 e boronic esters or the trimeric form of the boronic acids (boroxines) in solution.

122 sors are often based on fluorophore-appended boronic acids, but these severely lack discriminatory po

123 Starting from benzo-[b]-thiophene-2-boronic acid (BZB), a nanomolar inhibitor of AmpC beta-l

124 trabromopyrene and (4-(ethoxycarbonyl)phenyl)boronic acid can easily be coupled to prepare the requis

125 Pioneering work revealed that acyclic boronic acids can act as 'transition state analogue' inh

126 Here we show that boronic acids can be chemoselectively reacted in the pre

127 ow the interaction between carbohydrates and boronic acids can be combined with copper catalysis to a

128 Using the concept of boronic acid catalysis (BAC), electrophilic activation o

129 The efficacy of the new boronic acid catalyst was confirmed by its ability to ac

130 Alcohols can also be activated with boronic acid catalysts to form carbocation intermediates

131 In situ generation of boronic acid catechol ester derivatives generates RH(2)C

132 H3Hg(+) ensued a fast transmetalation of TPE-boronic acid causing drastic reduction in the solubility

133 phenols or benzoyl methyl hydroxamates, and boronic acid chemistries to reversibly join two [3-(1-ac

134 SX-517 is the first reported boronic acid chemokine antagonist and represents a novel

135 ng Pd-O-B linkages, a tri-coordinate (6-B-3) boronic acid complex and a tetra-coordinate (8-B-4) boro

136 adium-oxygen-boron linkages, a tricoordinate boronic acid complex, and two tetracoordinate boronate c

137 alized boronic acid to form a glucose-alkyne-boronic acid complex.

138 eboronation of polyfluoroaryl and heteroaryl boronic acids complicates their use in Suzuki-Miyaura co

139 s, provided 20 (VNRX-5133, taniborbactam), a boronic-acid-containing pan-spectrum beta-lactamase inhi

140 al engineering, where double-H-bonding donor boronic acids could act as suitable organocatalysts or t

141 ploys an air-stable diethanolamine-complexed boronic acid (DABO boronate) as the allyl transfer reage

142 eworks with compositions ranging from highly boronic acid-deficient to networks with catechol voids.

143 r molecule based on a 2-hydroxymethyl phenyl boronic acid derivative binds even at neutral pH to the

144 to electrophilic amination of several common boronic acid derivatives (e.g., pinacol esters).

145 A variety of aryl boronic acid derivatives and dialkylmalononitriles were

146 The reaction tolerates various boronic acid derivatives and functional groups.

147 ide starting materials with sp(2)-hybridized boronic acid derivatives and is compatible with heterocy

148 t synthesis of pyridine-based heteroaromatic boronic acid derivatives is reported through a novel dib

149 porphyrin and its Suzuki cross coupling with boronic acid derivatives.

150 reported efflux pump inhibitory activity of boronic acid derivatives.

151 e variation of the dye structure through the boronic acid derived moiety (approach (b)) enables the f

152 A series of boronic acid derived salicylidenehydrazone (BASHY) compl

153 thereby facilitating synthesis of the alkyl boronic acid drugs Velcade and Ninlaro as well as a boro

154 ient where one molecule was attracted to the boronic acid end of the gradient, and the other to the c

155 luoroboronate (FB(Ar(3))(-)) or an exogenous boronic acid/ester (ArB(OR)(2)) and nucleophilic activat

156 luorescein ditriflate with the electron-rich boronic acid/ester-functionalized pyrrole (2C/3C) and in

157 MIDA boronates (N-methylimidodiacetic boronic acid esters) serve as an increasingly general pl

158 Apart from this, boronic acids exhibit an exquisite reversible coordinati

159 While 2- and 4-substituted aryl boronic acids favored the (R)-enantiomer with most of th

160 rmolecular reductive C-N cross coupling with boronic acids, followed by intramolecular cyclization.

161 Large collections of chemically diverse boronic acid fragments are commercially available becaus

162 action is based on the rapid condensation of boronic acid functionalities with salicylhydroxamates.

163 trochemical cytosensor was designed based on boronic acid-functionalized polythiophene.

164 1-naphthaleneboronic acid and acenaphthene-5-boronic acid gave corresponding o-naphthyl benzaldehydes

165 functional groups, and should allow for the boronic acid group to be used as an effective traceless

166 y applicable for molecules with an intrinsic boronic acid group, but also for the other molecules tha

167 The use of a monomer bearing a boronic acid group, with its ability to specifically int

168 dation of BDBA resulted in the conversion of boronic acid groups to phenol groups.

169 ylation of gamma-vinyl-gamma-lactone by aryl boronic acid has been developed.

170 alkyl primary amines from the corresponding boronic acids has been achieved at ambient temperature m

171 ng reactivity of Au(III)-F species with aryl boronic acids has been studied in detail taking advantag

172 Boronic acids have attracted the attention of synthetic

173 of the current methods for the synthesis of boronic acids, however, require transition metal catalys

174 bjected to Pd-catalyzed Suzuki coupling with boronic acid in high yield.

175 kylboronic esters and the increasing role of boronic acids in drug discovery.

176 sociation constant (Ka) of ortho-substituted boronic acids in solution showed that Ka for 1:1 associa

177 In this review, the use of boronic acids in the construction of therapeutically use

178 tuted-3-iodoquinolin-4(1H)-ones with several boronic acids in water using Pd(OAc)2 as a catalyst and

179 ng-opening reaction of vinylcyclopropanes by boronic acids in water, using palladium nanoparticles fo

180 vaborbactam of the diazabicyclooctanone and boronic acid inhibitor classes, respectively, as new sca

181 virtual screening to produce nano-/picomolar boronic acid inhibitors of the carboxylesterase alphaE7

182 th the COF-1-type condensation of pyridine-4-boronic acid into a C(3) -symmetric trimeric boroxine mo

183 conversion of aryl, heteroaryl, and alkenyl boronic acids into sulfinate intermediates, and onwards

184 ve rapid and high-yielding conversion of the boronic acids into the corresponding sulfinates.

185 idate that the ipso amination of substituted boronic acids involves the formation of cyanamidyl/arylc

186 iented immobilization of antibodies in which boronic acid is directly attached to the surface and wit

187 When the boronic acid is ortho to the azo group, the thermodynami

188 ditions from both organotrifluoroborates and boronic acids is described.

189 -coupling between alkyl-carboxylic acids and boronic acids is described.

190 coupling of 1-aryl-2,2-difluoroalkenes with boronic acids is described.

191 lycal partners and diverse aryl- and alkenyl-boronic acids is presented, leading to original 2-ketogl

192 f heteroatom nucleophiles, O-alkylation with boronic acids is rare.

193 nes and barbituric acids, respectively, with boronic acids is reported.

194 its nitrile-N center with boron atom of the boronic acids, leading to chemoselective primary aminati

195 for aqueous-organic protodeboronation of 18 boronic acids, many widely viewed as unstable, have been

196 We have developed a synthetic boronic acid mask that restrains the ribonucleolytic act

197 Key synthetic transformations include phenyl boronic acid-mediated 6pai-electrocyclization reaction,

198 ol chemiluminescence (CL) biosensor based on boronic acid modified gold substrate has been developed

199 The boronic acid moiety greatly accelerates the initial form

200 nsor, pnGFP, based on the incorporation of a boronic acid moiety into a circularly permuted green flu

201 is achieved by introduction of a C-terminal boronic acid moiety into dipeptidic inhibitors of the Zi

202 h conditions amenable to the presence of the boronic acid moiety which was considered important for t

203 nd light conditions show that pai-conjugated boronic acid molecules are more effective crosslinkers o

204 exahydroxytriphenylene and 1,4-phenylene bis(boronic acid) monomers in solution.

205 edictions that more reactive warheads (e.g., boronic acids) must be employed to inhibit FAP than for

206 preparation of reactive allylic and benzylic boronic acids, obtained by reacting flow-generated diazo

207 ween alpha-hydroxycarboxylate of citrate and boronic acids of BDBA.

208 lene glycol polymers end-functionalized with boronic acids of varied structure to produce extensible

209 llowed expedient preparations of alpha-amino boronic acids, often with high stereoselectivity, thereb

210 show that the suppressive effect of peptide boronic acids on hyperactive Wnt signaling is dependent

211 ent, the imino group that forms ortho to the boronic acid or boronate ester group can form a dative N

212 N-tosylhydrazones, dihalogenated arenes, and boronic acids or boronate esters was developed, producin

213 with a range of aryl, heteroaryl, and styryl boronic acids or esters has been developed.

214 lyst to generate carbon radicals from either boronic acids or esters.

215 yl-Bpin, p-tolyl-Bcat) and the corresponding boronic acid (p-tolyl-B(OH)2) in this type of cross-coup

216 A wide range of sensitive boronic acids, particularly polyfluoroaryl substrates th

217 lexation of glucose and fructose with phenyl boronic acid (PBAc) followed by ethyl-acetate extraction

218 erine beta-lactamase inhibitors containing a boronic acid pharmacophore, with the goal of finding a p

219 However, aryl boronic acid pinacol (BPin) ester reagents can be diffic

220 presence of ostensibly equivalently reactive boronic acid pinacol (BPin) esters by kinetic discrimina

221 hese catalysts (CAL-3-Ir) can produce methyl boronic acid pinacol ester (CH(3) Bpin) in 29 % yield in

222 reactions from (S)-nicotine containing a C-4 boronic acid pinacol ester group.

223 inophenol and a Z- or an E-gamma-substituted boronic acid pinacol ester.

224 o organoboronic acids can also be applied to boronic acid pinacol esters and potassium organotrifluor

225 ction of commercial or readily accessed aryl boronic acid pinacol esters with alkyl lithium reagents

226 Alkenyl boronic acid pinacolates were found to be more suitable

227 d isocoumarins and 2-pyrones are isolated as boronic acids, pinacolboronate esters, or potassium orga

228 traceless protection of the C3/C5 diol with boronic acids prior to glycosylation.

229 n peroxide using hydropropidine and coumarin boronic acid probes, respectively.

230 Continuing the boronic acid program that led to vaborbactam, efforts we

231 tructure-activity analyses using a series of boronic acid proteasome inhibitors and correlate cytotox

232 onylative coupling of phthalimides with aryl boronic acids provides ready access to a broad range of

233 ent coupling of Selectfluor, a styrene and a boronic acid, provides chiral monofluorinated compounds

234 Condensation of oximes with boronic acids RB(OH)2 or B(OH)3 affords remarkably stabl

235 ted using a SNAP-tag approach to install the boronic acid reagent onto the extracellular domain of th

236 We repurposed the approximately 650 boronic acid reagents in our collection as a directed fr

237 An array of three water-soluble boronic acid receptors in combination with (19)F NMR spe

238 d on a quinolone fluorophore incorporating a boronic acid recognition element that gives it high affi

239 eptor pair and (b) functional tuning via the boronic acid residue.

240 Non-ortho-substituted boronic acids result in "flat" complexes.

241 died catalysts, meta-alkoxy substituted aryl boronic acids resulted in the (S)-enantiomer when used i

242 A ferrocenium boronic acid salt activates allylic alcohols to generate

243 2,6-Dimethoxy azobenzene boronic acids show an over 20-fold enhancement in bindin

244 nnectivity between the indole moiety and the boronic acid showed that, in particular, connectivity ex

245 rol experiments in the presence of competing boronic acids showed no crossover side-products and conf

246 are crosslinked with alkyl or pai-conjugated boronic acid small molecules (-B(OH)(2) ).

247 Control of boronic acid speciation is presented as a strategy to ac

248 e including the final trapping of a reactive boronic acid species with an aldehyde to generate a rang

249 a data set in which both the phosphoric and boronic acid structures were systematically varied, key

250 to an aryl ketone or aldehyde with an ortho-boronic acid substituent.

251 ween vicinal hydroxyl groups of arabitol and boronic acid substituents of the bithiophene functional

252 ithiophene) derivatives bearing cytosine and boronic acid substituents, in the presence of the inosin

253 Herein, we report on boronic acid-substituted stilbenes that limit TTR amyloi

254 ctions of benzylic alcohols, including other boronic acids such as 2,3,4,5-tetrafluorophenylboronic a

255 BL detection by the CLSI disk test (CLSI), a boronic acid-supplemented CLSI disk test (CLSI plus BA),

256 Boronic acid-supplemented tests can enhance ESBL detecti

257 ity exceeding 95%, with the exception of the boronic acid synergy test (88%) and modified Hodge test

258 ohort, sensitivities ranged from 72% for the boronic acid synergy test for the detection of KPC produ

259 arba assay, the Modified Carba NP assay, the boronic acid synergy test, and the metallo-beta-lactamas

260 ow protodeboronation, as do 3- and 4-pyridyl boronic acids (t0.5 > 1 week, pH 12, 70 degrees C).

261 DD.AA-type complexes of a series of aromatic boronic acids that adopt a syn-syn conformation with sui

262 We report a series of azobenzene boronic acids that reversibly control the extent of diol

263 up that lowers the pK(a) of the neighbouring boronic acid thereby facilitating diol binding at neutra

264 e other molecules that can be linked to aryl boronic acids through a self-immolative linker.

265 s and (ii) sequential disproportionations of boronic acid to borinic acid and borane.

266 ondary binding with an alkyne-functionalized boronic acid to form a glucose-alkyne-boronic acid compl

267 tal-free coupling of a tosyl hydrazone and a boronic acid to the preparation of a complex natural pro

268 epared through Rh-catalyzed addition of aryl boronic acids to 2,2-disubstituted malononitriles.

269 action tolerates a variety of functionalized boronic acids to afford a cis-fused bicyclic framework c

270 o-enol esters were subsequently coupled with boronic acids to afford tetrasubstituted alkene derivati

271 To this end, the ability of boronic acids to form reversible covalent bonds with hyd

272 the peculiar dynamic covalent reactivity of boronic acids to form tetraboronate derivatives, interes

273 lysed Csp(3) Suzuki coupling of acetals with boronic acids to generate benzylic ethers, a reaction th

274 unanimously in the related addition of aryl boronic acids to methacrylate derivatives.

275 nd stereoinvertive transmetalation of Csp(3) boronic acids to Pd(II).

276 ge of alkyl boronic esters and aryl or alkyl boronic acids to react with electron-deficient olefins v

277 OF-5 structure can form over a wide range of boronic acid-to-catechol ratios, thus producing framewor

278 arged dye molecules was demonstrated using a boronic acid-to-cationic gradient where one molecule was

279 ium-catalyzed carbonylative coupling of aryl boronic acids together with terminal alkynes and perfluo

280 Boronic acid transition-state inhibitors (BATSIs) repres

281 ation of 2-carbonyl-3-propargyl indoles with boronic acids under sequential palladium/triflic acid ca

282 In contrast, 2-pyridyl and 5-thiazolyl boronic acids undergo rapid protodeboronation (t0.5 appr

283 Cyclopropyl and vinyl boronic acids undergo very slow protodeboronation, as do

284 timal conditions for the slow release of the boronic acid using KOH as the base in biphasic THF/water

285 ere included in the investigations with each boronic acid varying in the substituent at its 4-positio

286 acid drugs Velcade and Ninlaro as well as a boronic acid version of the iconic antibiotic vancomycin

287 for the interconversion of diverse protected boronic acids, via intermediate organotrifluoroborates.

288 epatitis C virus (HCV), in which an N-benzyl boronic acid was essential for potent antiviral activity

289 th cytosine and bithiophene derivatized with boronic acid were used as functional monomers.

290 Boronic acids were investigated, and (31)P NMR binding e

291 irect benzylation between tosylhydrazone and boronic acid, which allowed the generation of structural

292 accharides can form tetrahedral adducts with boronic acids, which increases their nucleophilic charac

293 ling reactions involving aryl sulfamates and boronic acids, which operates at a significantly lower c

294 site-selective, copper-promoted couplings of boronic acids with carbohydrate derivatives.

295 described transnitrilative cyanation of aryl boronic acids with dialkylmalononitriles, the present re

296 This reaction is amenable to a wide range of boronic acids with different biorelevant functional grou

297 An efficient transnitrilation of aryl boronic acids with dimethylmalononitrile (DMMN) is descr

298 Condensation of boronic acids with hydroxyketones generates 1,3-dioxabor

299 Miyaura cross-coupling of unactivated Csp(3) boronic acids with perfect stereoretention.

300 endent, and varied substantially between the boronic acids, with rate maxima that varied over 6 order